Ibisobanuro
Insanganyamatsiko zacu zo muri Tofacitinib ni ingenzi mubikorwa byo gukora bya Tofacitinib, imiti izwi cyane ikoreshwa kugirango ifate ubwoko bumwe na bumwe bwa rubagimpande. Iri shyira hagati rifite uruhare runini mugukora urubyaro, zitanga umusanzu mubikorwa byacyo nubwiza. Binyuze muri (2r, 3r) -2,3-Bis [(4-methbenzoyl) aside ya succinique kandi - Igicuruzwa gisobanutse cya 3-1- (Igicuruzwa gisobanutse cya Synthesis gifite ubuziranenge bwa Tofacitibu.
Imiterere ya molekale nuburemere bwimikorere yacu ya tofacitinib byerekana ubuziranenge nubunini bwayo, bituma bigize igice cyizewe cyibikorwa bya farumasi. Hamwe nibikoresho byapimwe byitonze, iyi terambere ryizewe ko ihungabana nibikorwa byanyuma, tofacitinib. Ibintu byayo bya molekelar nabyo bigira uruhare mu kwikuramo muri rusange no ku buzima bwa filf, bukomeza kuba ingirakamaro kandi byizewe mu gihe kirekire.
Hitamo
Jdk afite ibikoresho byambere byitsinda ryakazi hamwe nibikoresho byo gucunga ubuziranenge, bizeza itangazo rihamye rya API hagati. Ikipe yabigize umwuga yizeza R & D ibicuruzwa. Kurwanya byombi, dushakisha CMO & CDMO mumasoko yo murugo kandi mpuzamahanga.