Ibisobanuro
Umuhuza wa Tokirastat hagati ya 2-cyanoisonIotic acide, CYA No 161233-97-2. Iki gicuruzwa kizwi kandi n'andi mazina: 2-cyanopyrine-acide ya 1-kanseri, 2-cyamamare Imiterere ya molecular yiyi ngingo hagati ni c7h4n2o2 nuburemere bwa molekile ni 148.1189. Nibintu byingenzi muri synthesis ya Tokirastat (ibiyobyabwenge bikoreshwa mugufata Hyperririnemia mubarwayi ba Gout).
2-cyanoisonIcotinic acide igira uruhare runini mu musaruro wa Tokirastat, ikora mu kubuza xanthine okidase, enzyme yagize uruhare mu musaruro uric. Nkigisubizo, urwego rutic aside mu maraso rugabanuka, kugabanya ibimenyetso by'abarwayi ba goutte. Iki kigo kimurika ni ikintu cyingenzi muburyo bwo gukora kuri Topirastat, bikaba igice cyibikorwa byinganda za farumasi.
Hitamo
Jdk afite ibikoresho byambere byitsinda ryakazi hamwe nibikoresho byo gucunga ubuziranenge, bizeza itangazo rihamye rya API hagati. Ikipe yabigize umwuga yizeza R & D ibicuruzwa. Kurwanya byombi, dushakisha CMO & CDMO mumasoko yo murugo kandi mpuzamahanga.