Tsanangudzo
Iyo molecular formula yeiyi yepakati ndeye C13H10CLN3O2s, uye uremu hwayo hwemanyorerwe 307.755. Yayo chaiyo molecular chimiro chinogonesa iyo inoshanda uye yakakwirira-yekuchena kugadzirwa kwe tofacitinib. Naizvozvo, iyo tofacitinib intermediate 1,4-chloro-7-p-toluenesulfonyl-2,3-d] pyrimidine chinhu chakakosha muindasitiri yechibheneketi kuti iite kurapwa kunobudirira kwezvirwere zvequemmune.
Zvigadzirwa zvedu zvinogadzirwa uchishandisa State-of-iyo-iyo-art maitiro kuti ive nechokwadi chekumusoro uye kusawirirana. Isu tinonzwisisa kukosha kwekuve akavimbika uye kwakachena mumishonga yekugadzira mishonga, ndosaka takazvipira kuchengetedza zviyero zvakanyanyisa panguva yekugadzira maitiro. Yedu tofacitinib intermediate 1,4-chloro-7-p-toluenesulfonyl-2,3-d-2,3-d kugadzikana kwekuchena kwakaomarara, kutendera vatengi vedu kuti vafunge nezvekuvimbika kweshoko rakakura.
Sarudza US
Jidk ine nzvimbo dzekutanga-dzekirasi dzekugadzira uye mhando dzemhando dzekutonga, dzinovimbisa kuwanikwa kwakagadzikana kweAPI vakapindirana. Nyanzvi yechikwata chivimbiso r & d yechigadzirwa. Kupesana nezvose zviri zviviri, tiri kutsvaga cmo & cdmo mumusika wemba uye wepasi rose.