Tsanangudzo
Topirastast Intermediate 2-Cyanoisonicotinic acid, Cas No. 161233-97-2. Ichi chigadzirwa chinozivikanwa zvakare nemamwe mazita: 2-Cyanopyridine-4-carboxyylic acid, 2-cyano-4-pyridinecarboycory acid, uye 4-pidridinecarboxy acid, 2-cyano-. Iyo molecular formula yeiyi yepakati compound ndeye c7h4n2o2 uye iyo molecular uremu ndeye 148.1189. Icho chinhu chakakosha mu synthesis yeTopirastast (mushonga unoshandiswa kurapa hyperuricemia mune gout varwere).
2-Cyanoiskucotinic Acid inodhura chiitiko chakakosha mukugadzirwa kweTopirasat, iyo inoshanda nekunyadzisa Xanthine oxidase, enzyme inobatanidzwa mukugadzirwa kweuric. Semhedzisiro, uric acid mazinga muropa kuderera, kusunungura zviratidzo zveGout varwere. Ichi chikamu chepakati chikamu chakakosha mune yekugadzira maitiro ePepirastast, ichiita kuti ive chikamu chakakosha cheindasitiri yemishonga yemishonga.
Sarudza US
Jidk ine nzvimbo dzekutanga-dzekirasi dzekugadzira uye mhando dzemhando dzekutonga, dzinovimbisa kuwanikwa kwakagadzikana kweAPI vakapindirana. Nyanzvi yechikwata chivimbiso r & d yechigadzirwa. Kupesana nezvose zviri zviviri, tiri kutsvaga cmo & cdmo mumusika wemba uye wepasi rose.