Sifo
Qaaciddada molika-ka ee dhexdhexaadka ah waa C13h10Cln3SO2s, iyo culeyska molecular waa 307.755. Qaab dhismeedka molicical ee saxda ah wuxuu awood u siinayaa soosaarka wax ku oolka ah iyo saadka-sareeya ee tofacitinib. Sidaa darteed, the toofatinitigister 1,4-chloro-7-p-toluenesulus-7h pyrrolo [2,3-d] Pyrrolo [2,3-d] Pyrroline [2,3-D] Pyrimidine waa qayb muhiim ah warshadaha dawooyinka si loo helo daaweyn wax ku ool ah oo loogu talagalay cudurrada iswada.
Alaabooyinkayaga waxaa loo soo saaray iyadoo la adeegsanayo hanaan-farshaxan-farshaxan si loo hubiyo tayada ugu sarreysa iyo joogteynta. Waxaan fahamsanahay muhiimadda ay leedahay in la isku halleyn karo oo ah waxsoosaarka daawooyinka ee dawooyinka, waana sababtaasna loogu heellan yahay joogteynta heerarka ugu adag inta lagu gudajiro howlaheena wax soo saarka. Tofacitibinif-ga Dhexe 1,4-chloro-7-p-toluenesulus-7h pyrrolo [2,3-d] pyrrolo [2,3-d] pyrroline [2,3-d] Pyrotine [2,3-d] Pyrotine [2,3-d] Pyrimidine-2,3-d] Pyrromine-ka [2,3-D] Pyrimidine-ka ayaa maraya daahir adag, deganaansho iyo imtixaanka nabadgelyada si loogu kalsoonaado ku kalsoon isku-darka murqaha ballaaran ee tofacitinib.
Na xulo
JDK wuxuu leeyahay tas-hiilaadka soosaarka ee fasalka iyo qalabka tayada tayada leh, taas oo xaqiijineysa sahayda xasilloonida ee API-da. Kooxda xirfadleyda ah ayaa xaqiijinaya R & D ee sheyga. Labadaba labadoodaba, waxaan raadineynaa CMO & CDMO suuqyada gudaha iyo kuwa caalamiga ah.